(E)-2-(2,3-Dichlorobenzylidene)hydrazine-1-carboximidamide acetate
Raphin1 acetate
CAS: 2242616-04-0
Molecular Formula: C10H12Cl2N4O2
(E)-2-(2,3-Dichlorobenzylidene)hydrazine-1-carboximidamide acetate - Names and Identifiers
| Name | Raphin1 acetate |
| Synonyms | Raphin1 acetate RAPHIN1 ACETATE (E)-2-(2,3-Dichlorobenzylidene)hydrazine-1-carboximidamide acetate |
| CAS | 2242616-04-0 |
(E)-2-(2,3-Dichlorobenzylidene)hydrazine-1-carboximidamide acetate - Physico-chemical Properties
| Molecular Formula | C10H12Cl2N4O2 |
| Molar Mass | 291.13 |
(E)-2-(2,3-Dichlorobenzylidene)hydrazine-1-carboximidamide acetate - References
| biological activity | Raphin1 acetate is a selective inhibitor of the orally bioavailable phospho-regulatory enzyme PPP1R15B (R15B). Raphin1 acetate can be tightly bound to R15B-PP1c holophorsphatase, corresponding to a Kd value of 0.033 μm. |
| Target | Value |
| R15B-PP1c (Cell-free assay) | 0.033 μM(Kd) |
Last Update：2024-04-09 20:49:11
